All Categories

Novel allosteric agonist of Sphingosine 1-phosphate receptor 2 (S1PR2)

GalR2-positive allosteric modulator

Antagonist for G-protein Coupled Receptor 7 (GPR7)

Novel mu;-δ opioid receptor heteromer-biased agonist with antinociceptive activity

Novel S1P1 agonist that does not require S1P-like headgroup interactions

An ATP-competitive small molecule that potently inhibits JAK1 and JAK2 kinases

Alkaloids

Alkaloids

Alkaloids

The first naturally occurring agonist for nuclear orphan receptor Nur77

An inhibitor of leucine-rich repeat kinase 2 (LRRK2; IC50s = 1.28 and 1.85 nM for wild-type and G2019S mutant forms of LRRK2, respectively)

Selective inhibitor of PI3Kγ-dependent Th17 cell differentiation

Refine Search