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Mps1-IN-2

Novel Mps1 inhibitor

Mps1-IN-3

Novel Potent and Selective MPS1 Inhibitor

MPT0B014

Novel inducer of G2/M arrest with down-regulation of Cdc (Tyr15) and Cdc25C, and up-regulation of cyclin B1, phospho-Cdc2 (Thr161) and Aurora A/B

MRL-871

Novel RORγt inhibitor, binding to a previously unidentified allosteric pocket in the RORγt LBD

MRS-1191

Selective A3 adenosine receptor antagonist

MRS-1754

Selective adenosine A2B receptor antagonist

MRT-10

Smoothened (Smo) receptor antagonist

MRT-83

A novel potent antagonist of SMO

MRT68921

Potent inhibitor of ULK1 and ULK2 in vitro, blocking autophagy in cells.

MS-275

A synthetic inhibitor of histone deacetylase (HDAC)

MS37452

Novel Modulator of Methyl-Lysine, inducing transcriptional derepression of p16/CDKN2A by disrupting CBX7ChD binding to H3K27me3 at the INK4A/ARF locus in PC3 prostate cancer cells.

MS436

Potent and selective BRD4 bromodomain inhibitor