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Selective Transient receptor potential vanilloid 4 (TRPV4) antagonist

A highly potent and orally bioavailable ATP-competitive inhibitor of PI3K and mTOR

Selective and orally active blocker of transient receptor potential vanilloid 4 (TRPV4)

A highly specific and potent inhibitor of PDK1 (3-Phosphoinositide dependent protein kinase-1)

A selective PDE4B(equal affinity to isoforms A-D) inhibitor.

Potent leucine-rich repeat kinase 2 (LRRK2) inhibitor

An orally available, potent, and selective PERK inhibitor

An orally bioavailable PI3K beta isoform-selective inhibitor

Bromodomain-containing proteins whose biological function is believed to function similarly to ACF1, the Drosophila BAZ2B ortholog

The first orally active, allosteric inhibitor of Wip1 phosphatase through flap-subdomain interaction

Novel human immune virus (HIV) maturation inhibitor

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