All Categories

A potent and selective Aurora A inhibitor with IC50 of 0.6 nM, more than 450-fold selectivity for Aurora A over Aurora B

Non-peptide, melanocortin MC receptor antagonist

Selective myosin light chain kinase inhibitor

Inhibitor of steroidogenic factor 1 (SF-1); Inverse agonists of the retinoic acid receptor (NR1B)

Inhibitor of steroidogenic factor 1 (SF-1); Inverse agonists of the retinoic acid receptor (NR1B)

Novel FKBP12 inhibitor

Highly potent inhibitor of the NF-kB pathway

Potent inhibitor of PDE4

The first small molecule, S1P2 selective agonist reported

Inhibitor of Staphylococcus Aureus Virulence; Non-competitive inhibitor of xanthine oxidase; Potent inhibitor of CYP2C9.

Inhibitor of DNA Polymerase III Holoenzyme System, Primase

Refine Search